Binding modes of CCR5-targetting HIV entry inhibitors: Partial and full antagonists
نویسندگان
چکیده
منابع مشابه
CCR5 Inhibitors and HIV
In August of 2007, the Food and Drug Administration (fda) approved the first chemokine (c-c motif) receptor 5 (ccr5) inhibitor, maraviroc, for treatment-experienced patients infected with r5-using virus. In an effort to better educate physicians and patients about these new drugs, this article will review the available clinical data on ccr5 antagonists and discuss implications for clinical prac...
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ژورنال
عنوان ژورنال: Journal of Molecular Graphics and Modelling
سال: 2008
ISSN: 1093-3263
DOI: 10.1016/j.jmgm.2007.12.003